ES412813A1 - Un procedimiento de preparacion de derivados de 1,2-benzoi-soxazol 3-sustituidos. - Google Patents

Un procedimiento de preparacion de derivados de 1,2-benzoi-soxazol 3-sustituidos.

Info

Publication number
ES412813A1
ES412813A1 ES412813A ES412813A ES412813A1 ES 412813 A1 ES412813 A1 ES 412813A1 ES 412813 A ES412813 A ES 412813A ES 412813 A ES412813 A ES 412813A ES 412813 A1 ES412813 A1 ES 412813A1
Authority
ES
Spain
Prior art keywords
substituted
soxazole
benzoi
derivatives
procedure
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES412813A
Other languages
English (en)
Spanish (es)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sumitomo Pharma Co Ltd
Original Assignee
Dainippon Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP2786672A external-priority patent/JPS5616154B2/ja
Priority claimed from JP2786572A external-priority patent/JPS5545545B2/ja
Application filed by Dainippon Pharmaceutical Co Ltd filed Critical Dainippon Pharmaceutical Co Ltd
Publication of ES412813A1 publication Critical patent/ES412813A1/es
Expired legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/20—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings condensed with carbocyclic rings or ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
ES412813A 1972-03-17 1973-03-17 Un procedimiento de preparacion de derivados de 1,2-benzoi-soxazol 3-sustituidos. Expired ES412813A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2786672A JPS5616154B2 (en]) 1972-03-17 1972-03-17
JP2786572A JPS5545545B2 (en]) 1972-03-17 1972-03-17

Publications (1)

Publication Number Publication Date
ES412813A1 true ES412813A1 (es) 1976-07-01

Family

ID=26365855

Family Applications (1)

Application Number Title Priority Date Filing Date
ES412813A Expired ES412813A1 (es) 1972-03-17 1973-03-17 Un procedimiento de preparacion de derivados de 1,2-benzoi-soxazol 3-sustituidos.

Country Status (10)

Country Link
US (1) US3948928A (en])
AU (1) AU466970B2 (en])
CA (1) CA1025857A (en])
CH (1) CH577984A5 (en])
DK (1) DK140498B (en])
ES (1) ES412813A1 (en])
FR (1) FR2181831B1 (en])
GB (1) GB1416071A (en])
NL (1) NL168833C (en])
SE (1) SE381047B (en])

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4728662A (en) * 1977-11-21 1988-03-01 Hoechst-Roussel Pharmaceuticals Inc. 1,2-benzisoxazoloxyacetic acids and related compounds
US4673746A (en) * 1978-10-06 1987-06-16 Hoechst-Roussel Pharmaceuticals, Inc. 1,2-benzisoxazoloxyacetic acids and related compounds
US4610988A (en) * 1982-04-09 1986-09-09 Hoechst-Roussel Pharmaceuticals Inc. 1-[3-(6-fluoro-1,2-benzisoxazol-3-yl)propyl]-4-(substituted)piperazines useful for alleviating pain
US4609658A (en) * 1982-04-09 1986-09-02 Hoechst-Roussel Pharmaceuticals Inc. 1-[3-(6-fluoro-1,2-benzisoxazol-3-yl)propyl]-4-(substituted) piperazines useful for reducing blood pressure
US4536578A (en) * 1982-04-09 1985-08-20 Hoechst-Roussel Pharmaceuticals Inc. 1-[3-(6-Fluoro-1,2-benzisoxazol-3-yl)propyl]-4-(substituted)piperazines
JPS58201770A (ja) * 1982-05-18 1983-11-24 Dainippon Pharmaceut Co Ltd α−置換−１，２−ベンズイソキサゾ−ル−３−酢酸エステル類並びにその酸付加塩類及び第４級アンモニウム塩類
ATE398616T1 (de) * 2005-02-04 2008-07-15 Ctg Pharma S R L Neue 4-aminochinolinderivate als antimalariamittel
US8034953B2 (en) 2005-05-10 2011-10-11 Incyte Corporation Modulators of indoleamine 2,3-dioxygenase and methods of using the same
JP5294874B2 (ja) * 2005-12-20 2013-09-18 インサイト・コーポレイション インドールアミン２，３−ジオキシゲナーゼのモジュレーターとしてのｎ−ヒドロキシアミジノヘテロ環
WO2007081335A1 (en) * 2006-01-12 2007-07-19 Merck & Co., Inc. Therapeutic compounds for treating dyslipidemic conditions
WO2008036652A2 (en) * 2006-09-19 2008-03-27 Incyte Corporation Amidines as modulators of indoleamine 2,3-dioxygenase
CA2663057C (en) * 2006-09-19 2015-12-08 Incyte Corporation N-hydroxyamidinoheterocycles as modulators of indoleamine 2,3-dioxygenase
CL2007002650A1 (es) 2006-09-19 2008-02-08 Incyte Corp Compuestos derivados de heterociclo n-hidroxiamino; composicion farmaceutica, util para tratar cancer, infecciones virales y desordenes neurodegenerativos entre otras.
WO2008058178A1 (en) * 2006-11-08 2008-05-15 Incyte Corporation N-hydroxyamidinoheterocycles as modulators of indoleamine 2,3-dioxygenase
JP2010527965A (ja) * 2007-05-24 2010-08-19 ノイロサーチ アクティーゼルスカブ 例えば呼吸器疾患、てんかん及び痙攣の治療のためのカリウムチャネル調節剤としてのベンゾイソオキサゾール誘導体
MY192633A (en) 2008-07-08 2022-08-29 Incyte Holdings Corp 1,2,5-oxadiazoles as inhibitors of indoleamine 2,3-dioxygenase
EP3744715A1 (en) 2013-11-08 2020-12-02 Incyte Holdings Corporation Process for the synthesis of an indoleamine 2,3-dioxygenase inhibitor

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1670497C3 (de) * 1967-06-06 1973-12-20 Chinoin Gyogyszer- Es Vegyeszeti Termekek Gyara Rt, Budapest Isochinohnderivate und Verfahren zu deren Herstellung

Also Published As

Publication number Publication date
CH577984A5 (en]) 1976-07-30
AU5347973A (en) 1974-09-19
DK140498C (en]) 1980-03-17
GB1416071A (en) 1975-12-03
DK140498B (da) 1979-09-17
CA1025857A (en) 1978-02-07
NL168833C (nl) 1982-05-17
NL168833B (nl) 1981-12-16
SE381047B (sv) 1975-11-24
US3948928A (en) 1976-04-06
FR2181831A1 (en]) 1973-12-07
FR2181831B1 (en]) 1975-10-10
NL7303682A (en]) 1973-09-19
AU466970B2 (en) 1975-11-13

Similar Documents

Publication Publication Date Title
IE40046L (en) Benzimidazole derivatives
ES412813A1 (es) Un procedimiento de preparacion de derivados de 1,2-benzoi-soxazol 3-sustituidos.
BG25991A3 (bg) Метод за получаване на 1,2-бензизоксазолови производни
SE390819B (sv) Analogiforfarande for framstellning av piperazinyl-propyl-1,2,4-triazolinderivat
DK135454B (da) Analogifremgangsmåde til fremstilling af 2,1,3-benzothiadiazolderivater.
FI49503C (fi) Analogiamenetelmä 1,2,3,4-tetrahydro-4-fenyyli-isokinoliinijohdannaist en valmistamiseksi.
ES403445A1 (es) Procedimiento para la obtencion de derivados de la oxadia- zolona.
DK135505B (da) Analogifremgangsmåde til fremstilling af morpholinderivater.
DK134490B (da) Analogifremgangsmåde til fremstilling af 2,6-diaminonebularin-derivater.
SE393612B (sv) Forfarande for framstellning av vissa angivna benso-1,2,4-triazin-di-n-oxider
DK135991B (da) Analogifremgangsmåde til fremstilling af 2-oxazolinderivater.
ES428005A1 (es) Procedimiento para la preparacion de derivados de 3-4-dihi-dro-2h-naftalenom-(1)-5-oxi-propil-piperazina.
ES429871A1 (es) Procedimiento de preparacion de derivados 1, 3-benzodioxol.
FI52735C (fi) Menetelmä uusien pregnadieeni-21-happojohdannaisten valmistamiseksi.
ES421130A1 (es) Procedimiento para preparar derivados de ditiino (1,4) (2, 3-c) pirrol.
ES462849A1 (es) Un procedimiento para la preparacion de nuevos derivados de 3,5-diona-4,4-dimetil-pirrolidina.
SE401833B (sv) Forfarande for framstellnig av vissa angivna 1,2,4-friazolderivat
ES411710A1 (es) Procedimiento para la preparacion de nitroimidazolil-tria- zolo-piridazinas.
SE419980B (sv) Forfarande for framstellning av eventuellt substituerade 2-fenyl-bicyklo /2,2,2/okt-3-ylalkylaminer
SE418084B (sv) Forfarande for framstellning av 1,2,4-bensotiadiazin-derivat
ES436605A1 (es) Procedimiento para la preparacion de 3-(5-nitro-1-metil-2- imidazoli) -5-triazolon4, 3-bn piridazinas.
SE387636B (sv) Forfarande for framstellning av 2-substituerade 1,3,4- tiadiazol-5-tioler
SE383518B (sv) Forfarande for framstellning av derivat av 1,4-etano-2,3-dihydro-kinolin.
NO138140C (no) Fremgangsmaate for fremstilling av 4,4`-ditert.butyl-benzoylperoksyd
AR204011A1 (es) Procedimiento de preparacion de nuevos derivados de 7-h-indolizino(5,6,7-ij)isoquinoleina